{"id":69,"date":"2020-09-11T15:43:00","date_gmt":"2020-09-11T13:43:00","guid":{"rendered":"http:\/\/niemusibolec.com\/?p=69"},"modified":"2020-11-27T17:55:07","modified_gmt":"2020-11-27T16:55:07","slug":"jak-dziala-paracetamol","status":"publish","type":"post","link":"https:\/\/niemusibolec.com\/index.php\/2020\/09\/11\/jak-dziala-paracetamol\/","title":{"rendered":"Jak dzia\u0142a: paracetamol"},"content":{"rendered":"<p>[et_pb_section fb_built=&#8221;1&#8243; fullwidth=&#8221;on&#8221; next_background_color=&#8221;#f0b800&#8243; _builder_version=&#8221;4.0.4&#8243; bottom_divider_style=&#8221;slant&#8221; bottom_divider_flip=&#8221;horizontal&#8221;][et_pb_fullwidth_header title=&#8221;Paracetamol&#8221; subhead=&#8221;jak dzia\u0142a ten lek?&#8221; text_orientation=&#8221;center&#8221; background_overlay_color=&#8221;rgba(52,81,104,0.8)&#8221; _builder_version=&#8221;4.0.4&#8243; title_font=&#8221;Lato|700|||||||&#8221; title_font_size=&#8221;46px&#8221; title_line_height=&#8221;1.5em&#8221; content_font=&#8221;Lato||||||||&#8221; content_font_size=&#8221;20px&#8221; content_line_height=&#8221;1.8em&#8221; subhead_font=&#8221;Lato|700|||||||&#8221; subhead_font_size=&#8221;25px&#8221; subhead_line_height=&#8221;1.5em&#8221; background_color=&#8221;#afafaf&#8221; background_image=&#8221;httpss:\/\/niemusibolec.com\/wp-content\/uploads\/2020\/09\/christina-victoria-craft-ZHys6xN7sUE-unsplash-scaled.jpg&#8221; custom_margin=&#8221;|||&#8221; custom_padding=&#8221;5vw||150px||false&#8221; animation_style=&#8221;slide&#8221; animation_direction=&#8221;top&#8221; animation_intensity_slide=&#8221;2%&#8221; title_font_size_tablet=&#8221;36px&#8221; title_font_size_phone=&#8221;&#8221; title_font_size_last_edited=&#8221;on|phone&#8221; button_one_text_size__hover_enabled=&#8221;off&#8221; button_two_text_size__hover_enabled=&#8221;off&#8221; button_one_text_color__hover_enabled=&#8221;off&#8221; button_two_text_color__hover_enabled=&#8221;off&#8221; button_one_border_width__hover_enabled=&#8221;off&#8221; button_two_border_width__hover_enabled=&#8221;off&#8221; button_one_border_color__hover_enabled=&#8221;off&#8221; button_two_border_color__hover_enabled=&#8221;off&#8221; button_one_border_radius__hover_enabled=&#8221;off&#8221; button_two_border_radius__hover_enabled=&#8221;off&#8221; button_one_letter_spacing__hover_enabled=&#8221;off&#8221; button_two_letter_spacing__hover_enabled=&#8221;off&#8221; button_one_bg_color__hover_enabled=&#8221;off&#8221; button_two_bg_color__hover_enabled=&#8221;off&#8221;][\/et_pb_fullwidth_header][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; next_background_color=&#8221;#ffffff&#8221; admin_label=&#8221;Quote&#8221; _builder_version=&#8221;4.0.4&#8243; background_color=&#8221;#f0b800&#8243; custom_padding=&#8221;||150px||false&#8221; bottom_divider_style=&#8221;slant&#8221; bottom_divider_flip=&#8221;horizontal&#8221;][et_pb_row _builder_version=&#8221;4.0.4&#8243; width=&#8221;90%&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;3.25&#8243; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_text _builder_version=&#8221;4.0.4&#8243; text_font=&#8221;Farsan||||||||&#8221; text_text_color=&#8221;#ffffff&#8221; text_font_size=&#8221;27px&#8221; text_line_height=&#8221;1.5em&#8221; header_font=&#8221;||||||||&#8221; text_orientation=&#8221;center&#8221; max_width=&#8221;800px&#8221; module_alignment=&#8221;center&#8221; text_font_size_tablet=&#8221;36px&#8221; text_font_size_phone=&#8221;26px&#8221; text_font_size_last_edited=&#8221;on|desktop&#8221;]Zna go praktycznie ka\u017cdy &#8211; to jeden z lek\u00f3w przeciwb\u00f3lowych dost\u0119pnych bez recepty nie tylko w aptece, ale te\u017c praktycznie w ka\u017cdym sklepie, kiosku i na ka\u017cdej stacji benzynowej. Czy jednak wiesz, kiedy i w jaki spos\u00f3b go stosowa\u0107, aby by\u0142 bezpieczny i skuteczny?[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; next_background_color=&#8221;#f0b800&#8243; admin_label=&#8221;About Me&#8221; _builder_version=&#8221;3.22&#8243; background_color=&#8221;#ffffff&#8221; custom_padding=&#8221;||150px||false|false&#8221; bottom_divider_style=&#8221;slant&#8221; bottom_divider_flip=&#8221;horizontal&#8221;][et_pb_row _builder_version=&#8221;3.25&#8243;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;3.25&#8243; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_text _builder_version=&#8221;3.27.4&#8243; text_font=&#8221;Lato||||||||&#8221; text_font_size=&#8221;18px&#8221; text_line_height=&#8221;1.8em&#8221; link_font=&#8221;||||||||&#8221; ul_font=&#8221;||||||||&#8221; ol_font=&#8221;||||||||&#8221; quote_font=&#8221;||||||||&#8221; header_font=&#8221;||||||||&#8221; header_2_font=&#8221;Lato|700|||||||&#8221; header_2_font_size=&#8221;30px&#8221; header_2_letter_spacing=&#8221;1px&#8221; header_2_line_height=&#8221;1.5em&#8221; animation_style=&#8221;slide&#8221; animation_direction=&#8221;bottom&#8221; animation_intensity_slide=&#8221;5%&#8221; header_2_font_size_tablet=&#8221;&#8221; header_2_font_size_phone=&#8221;22px&#8221; header_2_font_size_last_edited=&#8221;on|phone&#8221;]Paracetamol (inna jego nazwa to acetaminofen) to lek o dzia\u0142aniu przeciwb\u00f3lowym i przeciwgor\u0105czkowym &#8211; tak w zasadzie zaczyna si\u0119 ka\u017cdy opis tej substancji, kt\u00f3ry znajdziecie w internecie. I to sama prawda! Ale z czego wynika to dzia\u0142anie i na czym w zasadzie polega? Aby to zrozumie\u0107, musimy troch\u0119 zag\u0142\u0119bi\u0107 si\u0119 w metabolizm ludzkiego organizmu &#8211; obiecuj\u0119, nie b\u0119dzie nudno!<\/p>\n<p>W naszym ciele wyst\u0119puj\u0105 ciekawe substancje nazywane prostaglandynami. Mamy ich kilkana\u015bcie r\u00f3\u017cnych rodzaj\u00f3w. To w zasadzie hormony &#8211; ale hormony parakrynowe, czyli takie, kt\u00f3re dzia\u0142aj\u0105 miejscowo &#8211; pomimo, \u017c\u0119 wydzielane s\u0105 r\u00f3wnie\u017c do krwi, to czas ich rozpadu jest po prostu bardzo kr\u00f3tki. Znajduj\u0105 si\u0119 we wszystkich tkankach i p\u0142ynach ustrojowych naszego organizmu&#8230; ale dlaczego w og\u00f3le s\u0105 wydzielane?<\/p>\n<p>Nasze tkanki produkuj\u0105 prostaglandyny w odpowiedzi na zadzia\u0142anie r\u00f3\u017cnych czynnik\u00f3w &#8211; nie tylko uszkadzaj\u0105cych (takich jak np. toksyny czy patogeny), ale r\u00f3wnie\u017c hormon\u00f3w czy neuroprzeka\u017anik\u00f3w. Dziwne? No dziwne. A jeszcze dziwniejsze jest to, \u017ce w zale\u017cno\u015bci od sytuacji prostaglandyny potrafi\u0105 zmusza\u0107 nasze tkanki&#8230; do przeciwstawnego dzia\u0142ania! Opr\u00f3cz najistotniejszego dla nas w dzisiejszych rozwa\u017caniach dzia\u0142ania, czyli bycia mediatorem procesu zapalnego (czyli jedn\u0105 z substancji ten proces zapalny wytwarzaj\u0105c\u0105) i np. pobudzania ruchliwo\u015bci plemnik\u00f3w, prostaglandyny na mi\u0119\u015bnie g\u0142adkie w naszym ciele dzia\u0142aj\u0105 albo pobudzaj\u0105c, albo hamuj\u0105c ich skurcze. Ot, takie dziwowisko &#8211; dzia\u0142aj\u0105 tak na mi\u0119\u015bni\u00f3wk\u0119 macicy, przewodu pokarmowego, uk\u0142adu oddechowego czy naczy\u0144 krwiono\u015bnych.<\/p>\n<p>Ale wr\u00f3\u0107my do paracetamolu. Paracetamol powoduje, \u017ce te prostaglandyny, kt\u00f3re mia\u0142yby zosta\u0107 wytworzone (wybaczcie, zsyntetyzowane tu trudne s\u0142owo, a ja zawsze sobie w g\u0142owie czytam&#8230; wiec wytworzone) w naszym o\u015brodkowym uk\u0142adzie nerwowym&#8230; nie powstan\u0105. Lek ten blokuje jeden z etap\u00f3w syntezy prostaglandyn, a to troch\u0119 jak z pieczeniem ciasta &#8211; je\u015bli dodacie do brownie wszystkie sk\u0142adniki, ale w\u0142o\u017cycie go do zimnego piekarnika&#8230; to raczej si\u0119 nie najecie \ud83d\ude09 Tutaj podobnie. Zablokowanie tego procesu wywo\u0142uje w\u0142a\u015bnie dzia\u0142anie przeciwb\u00f3lowe i przeciwgor\u0105czkowe, ale skoro dzia\u0142a tylko w OUN, a nie &#8222;na obwodzie&#8221; (czyli w ca\u0142ym organizmie), to nie mo\u017cemy oczekiwa\u0107 od paracetamolu np. dzia\u0142ania przeciwzapalnego po urazie kolana&#8230; ale jednocze\u015bnie paracetamol nie uszkadza b\u0142ony \u015bluzowej \u017co\u0142\u0105dka i nie ma wp\u0142ywu na krzepni\u0119cie krwi.[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; next_background_color=&#8221;#ffffff&#8221; admin_label=&#8221;Quote&#8221; _builder_version=&#8221;4.0.4&#8243; background_color=&#8221;#f0b800&#8243; custom_padding=&#8221;||150px||false&#8221; bottom_divider_style=&#8221;slant&#8221; bottom_divider_flip=&#8221;horizontal&#8221;][et_pb_row _builder_version=&#8221;4.0.4&#8243; width=&#8221;90%&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;3.25&#8243; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_text _builder_version=&#8221;4.0.4&#8243; text_font=&#8221;Farsan||||||||&#8221; text_text_color=&#8221;#ffffff&#8221; text_font_size=&#8221;27px&#8221; text_line_height=&#8221;1.5em&#8221; header_font=&#8221;||||||||&#8221; text_orientation=&#8221;center&#8221; max_width=&#8221;800px&#8221; module_alignment=&#8221;center&#8221; text_font_size_tablet=&#8221;36px&#8221; text_font_size_phone=&#8221;26px&#8221; text_font_size_last_edited=&#8221;on|desktop&#8221;]To wszystko sprawia, \u017ce mo\u017cemy \u015bmia\u0142o stwierdzi\u0107, \u017ce paracetamol jest bezpiecznym i skutecznym w wielu sytuacjach. Mo\u017cna go stosowa\u0107 r\u00f3wnie\u017c u kobiet w ci\u0105\u017cy i w trakcie laktacji (oczywi\u015bcie po uzgodnieniu z lekarzem) i u dzieci od 3-ego miesi\u0105ca \u017cycia.[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; next_background_color=&#8221;#f0b800&#8243; admin_label=&#8221;About Me&#8221; _builder_version=&#8221;3.22&#8243; background_color=&#8221;#ffffff&#8221; custom_padding=&#8221;||150px||false|false&#8221; bottom_divider_style=&#8221;slant&#8221; bottom_divider_flip=&#8221;horizontal&#8221;][et_pb_row _builder_version=&#8221;3.25&#8243;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;3.25&#8243; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_text _builder_version=&#8221;4.0.4&#8243; text_font=&#8221;Lato||||||||&#8221; text_font_size=&#8221;18px&#8221; text_line_height=&#8221;1.8em&#8221; link_font=&#8221;||||||||&#8221; ul_font=&#8221;||||||||&#8221; ol_font=&#8221;||||||||&#8221; quote_font=&#8221;||||||||&#8221; header_font=&#8221;||||||||&#8221; header_2_font=&#8221;Lato|700|||||||&#8221; header_2_font_size=&#8221;30px&#8221; header_2_letter_spacing=&#8221;1px&#8221; header_2_line_height=&#8221;1.5em&#8221; animation_style=&#8221;slide&#8221; animation_direction=&#8221;bottom&#8221; animation_intensity_slide=&#8221;5%&#8221; header_2_font_size_tablet=&#8221;&#8221; header_2_font_size_phone=&#8221;22px&#8221; header_2_font_size_last_edited=&#8221;on|phone&#8221;]<\/p>\n<p>Paracetamol jest lekiem metabolizowanym w w\u0105trobie &#8211; oznacza to, \u017ce nasz organizm rozk\u0142ada go w\u0142a\u015bnie w tym narz\u0105dzie. To istotna informacja, bo podstawowym przeciwwskazaniem do jego stosowania jest w\u0142a\u015bnie ci\u0119\u017cka niewydolno\u015b\u0107 w\u0105troby (a tak\u017ce inne choroby metaboliczne upo\u015bledzaj\u0105ce jej dzia\u0142anie, odwodnienie, ci\u0119\u017ckie niedo\u017cywienie lub choroba alkoholowa). Do tego wszystkiego przedawkowanie paracetamolu uszkadza najbardziej w\u0142a\u015bnie w\u0105trob\u0119 &#8211; przyj\u0119cie dwukrotno\u015bci dziennej dawki maksymalnej mo\u017ce spowodowa\u0107 trwa\u0142e uszkodzenie w\u0105troby. Mamy oczywi\u015bcie na paracetamol odtrutk\u0119, ale pomoc musi przyj\u015b\u0107 szybko.<\/p>\n<p>W leczeniu b\u00f3lu ostrego paracetamol jest chyba najcz\u0119\u015bciej stosowany w przypadku b\u00f3lu g\u0142owy czy gor\u0105czki &#8211; i jest w tych sytuacjach bardzo skuteczny. Je\u015bli chodzi o b\u00f3l przewlek\u0142y, to paracetamol rzadko bywa stosowany jako jedyny lek, jednak bardzo cz\u0119sto wykorzystujemy go \u0142\u0105cz\u0105c z innymi lekami przeciwb\u00f3lowymi. Takie post\u0119powanie umo\u017cliwia nam osi\u0105gni\u0119cie lepszego efektu przy zastosowaniu mniejszych dawek poszczeg\u00f3lnych lek\u00f3w (ka\u017cdy z nich ma inny mechanizm dzia\u0142ania, wi\u0119c wp\u0142ywa na r\u00f3\u017cne elementy z ca\u0142ego szlaku przewodzenia b\u00f3lu (<a href=\"httpss:\/\/niemusibolec.com\/index.php\/2020\/09\/10\/8\/\">a jak taki szlak dla b\u00f3lu receptorowego wygl\u0105da przeczytasz tu<\/a>) &#8211; dzi\u0119ki temu hamowanie odczuwania b\u00f3lu jest skuteczniejsze, ni\u017c gdyby\u015bmy u\u017cyli tylko jednego leku).<\/p>\n<p>Jak stosowa\u0107 paracetamol?<\/p>\n<p>[\/et_pb_text][et_pb_blurb title=&#8221;przede wszystkim adekwatnie do sytuacji &#8211; to dobry lek na b\u00f3l g\u0142owy czy gor\u0105czk\u0119, ale s\u0142aby do stosowania samodzielnego np. przy urazie stawu (przez brak dzia\u0142ania przeciwzapalnego);&#8221; use_icon=&#8221;on&#8221; font_icon=&#8221;%%202%%&#8221; icon_color=&#8221;#ffb356&#8243; icon_placement=&#8221;left&#8221; content_max_width=&#8221;1100px&#8221; use_icon_font_size=&#8221;on&#8221; icon_font_size=&#8221;22px&#8221; _builder_version=&#8221;4.0.4&#8243; header_font=&#8221;Lato|700|||||||&#8221; header_font_size=&#8221;16px&#8221; header_line_height=&#8221;1.4em&#8221; body_font=&#8221;||||||||&#8221; custom_margin=&#8221;|||&#8221; animation_style=&#8221;slide&#8221; animation_direction=&#8221;bottom&#8221; animation_intensity_slide=&#8221;5%&#8221; locked=&#8221;off&#8221;][\/et_pb_blurb][et_pb_blurb title=&#8221;zgodnie z jego farmakokinetyk\u0105: pojedyncza dawka paracetamolu dzia\u0142a 4-6 godzin, wi\u0119c je\u015bli stosujemy go w b\u00f3lu przewlek\u0142ym (bez konsultacji z lekarzem mo\u017cna stosowa\u0107 go na b\u00f3l maksymalnie 10 dni, na gor\u0105czk\u0119 &#8211; 3 dni) powinni\u015bmy go stosowa\u0107 w\u0142a\u015bnie w tym rytmie aby by\u0142 skuteczny;&#8221; use_icon=&#8221;on&#8221; font_icon=&#8221;%%202%%&#8221; icon_color=&#8221;#ffb356&#8243; icon_placement=&#8221;left&#8221; content_max_width=&#8221;1100px&#8221; use_icon_font_size=&#8221;on&#8221; icon_font_size=&#8221;22px&#8221; _builder_version=&#8221;4.0.4&#8243; header_font=&#8221;Lato|700|||||||&#8221; header_font_size=&#8221;16px&#8221; header_line_height=&#8221;1.4em&#8221; body_font=&#8221;||||||||&#8221; custom_margin=&#8221;|||&#8221; animation_style=&#8221;slide&#8221; animation_direction=&#8221;bottom&#8221; animation_intensity_slide=&#8221;5%&#8221; locked=&#8221;off&#8221;][\/et_pb_blurb][et_pb_blurb title=&#8221;zgodnie z jego dawkowaniem: dla doros\u0142ego pojedyncza dawka to od 300 do 1000mg, w zale\u017cno\u015bci od tego, jak cz\u0119sto go przyjmujemy; maksymalna dawka dobowa nie powinna przekracza\u0107 4g (a je\u015bli stosujemy go kilka dni pod rz\u0105d &#8211; to 2,5g); to dawkowanie dotyczy doros\u0142ego, zdrowego cz\u0142owieka &#8211; w przypadku np. dzieci musi by\u0107 zmodyfikowane zgodnie z zaleceniami lekarza prowadz\u0105cego;&#8221; use_icon=&#8221;on&#8221; font_icon=&#8221;%%202%%&#8221; icon_color=&#8221;#ffb356&#8243; icon_placement=&#8221;left&#8221; content_max_width=&#8221;1100px&#8221; use_icon_font_size=&#8221;on&#8221; icon_font_size=&#8221;22px&#8221; _builder_version=&#8221;4.0.4&#8243; header_font=&#8221;Lato|700|||||||&#8221; header_font_size=&#8221;16px&#8221; header_line_height=&#8221;1.4em&#8221; body_font=&#8221;||||||||&#8221; custom_margin=&#8221;|||&#8221; animation_style=&#8221;slide&#8221; animation_direction=&#8221;bottom&#8221; animation_intensity_slide=&#8221;5%&#8221; locked=&#8221;off&#8221;][\/et_pb_blurb][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; next_background_color=&#8221;#ffffff&#8221; admin_label=&#8221;Quote&#8221; _builder_version=&#8221;4.0.4&#8243; background_color=&#8221;#f0b800&#8243; custom_padding=&#8221;||150px||false&#8221; bottom_divider_style=&#8221;slant&#8221; bottom_divider_flip=&#8221;horizontal&#8221;][et_pb_row _builder_version=&#8221;4.0.4&#8243; width=&#8221;90%&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;3.25&#8243; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_text _builder_version=&#8221;4.0.4&#8243; text_font=&#8221;Farsan||||||||&#8221; text_text_color=&#8221;#ffffff&#8221; text_font_size=&#8221;27px&#8221; text_line_height=&#8221;1.5em&#8221; header_font=&#8221;||||||||&#8221; text_orientation=&#8221;center&#8221; max_width=&#8221;800px&#8221; module_alignment=&#8221;center&#8221; text_font_size_tablet=&#8221;36px&#8221; text_font_size_phone=&#8221;26px&#8221; text_font_size_last_edited=&#8221;on|desktop&#8221;]Stosuj\u0105c paracetamol &#8211; szczeg\u00f3lnie w przypadku gor\u0105czki w przebiegu infekcji wirusowych &#8211; zachowaj ostro\u017cno\u015b\u0107. Wiele lek\u00f3w &#8222;na przezi\u0119bienie&#8221; (na temat u\u017cywania kt\u00f3rych jako leczenia przezi\u0119bienia mam osobiste negatywne zdanie, ale mo\u017ce o tym kiedy indziej) zawiera w swoim sk\u0142adzie w\u0142a\u015bnie t\u0105 substancj\u0119. Czytaj sk\u0142ady lek\u00f3w, kt\u00f3re ze sob\u0105 \u0142\u0105czysz, aby nie przekroczy\u0107 dobowej dawki maksymalnej paracetamolu (i innych substancji).[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section]<\/p>\n","protected":false},"excerpt":{"rendered":"<p>[et_pb_section fb_built=&#8221;1&#8243; fullwidth=&#8221;on&#8221; next_background_color=&#8221;#f0b800&#8243; _builder_version=&#8221;4.0.4&#8243; bottom_divider_style=&#8221;slant&#8221; bottom_divider_flip=&#8221;horizontal&#8221;][et_pb_fullwidth_header title=&#8221;Paracetamol&#8221; subhead=&#8221;jak dzia\u0142a ten lek?&#8221; text_orientation=&#8221;center&#8221; background_overlay_color=&#8221;rgba(52,81,104,0.8)&#8221; _builder_version=&#8221;4.0.4&#8243; title_font=&#8221;Lato|700|||||||&#8221; title_font_size=&#8221;46px&#8221; title_line_height=&#8221;1.5em&#8221; content_font=&#8221;Lato||||||||&#8221; content_font_size=&#8221;20px&#8221; content_line_height=&#8221;1.8em&#8221; 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